RAS Chemistry & Material ScienceЖурнал общей химии Russian Journal of General Chemistry

  • ISSN (Print) 0044-460X
  • ISSN (Online) 3034-5596

Synthesis, luminescent properties and antibacterial activity of new pyrazoline and pyrimidine derivatives of (2e)-1-biphenyl-3-arylprop-2-en-1-ones

PII
10.31857/S0044460X23090032-1
DOI
10.31857/S0044460X23090032
Publication type
Article
Status
Published
Authors
Volume/ Edition
Volume 93 / Issue number 9
Pages
1335-1342
Abstract
Substituted prop-2-en-1-ones were obtained by the condensation reaction of 1-biphenyl-4-yl-ethanone with aromatic aldehydes in the presence of sodium hydroxide in an aqueous ethanol solution. Subsequent cyclization of the latter with hydrazine hydrate, phenylhydrazine, and thiosemicarbazide in an acidic medium leads to the corresponding pyrazolines. The reaction of amidine hydrochlorides with chalcones in a KOH-ethanol system leads to 2,4,6-trisubstituted pyrimidines. The luminescent and antibacterial properties of the resulting systems was studied.
Keywords
замещенные проп-2-ен-1-оны люминесценсия пиразолины пиримидины гетероциклизация антибактериальная активность
Date of publication
15.09.2023
Year of publication
2023
Number of purchasers
0
Views
33

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